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Huwentoxin-XVI

簡要描述:Smartox Biotechnology是*一家專門生產(chǎn)動(dòng)物毒液多肽毒素,用于細(xì)胞離子通道功能研究的生物醫(yī)藥公司。多肽毒素在生物制藥領(lǐng)域具有重要的使用價(jià)值。

  • 產(chǎn)品型號:
  • 廠商性質(zhì):代理商
  • 更新時(shí)間:2024-08-27
  • 訪  問  量:1446

產(chǎn)品介紹

Huwentoxin-XVI

Huwentoxin-XVI is a selective blocker of N-type Ca2+channels

NCa2+通道選擇性阻斷劑

 is a 39 amino acids peptide that was discovered from the venom of the Chinese tarantula Ornithoctonus huwena was shown to be a potent blocker of HVA N-type calcium channels with an IC50 value of 60 nM in rat DRG. The blocking effect appears to be similar to that of  ω-conotoxin-GVIA and ω-conotoxin-MVIIA. Neverthelss,  differs from GVIA and MVIIA thanks to its greater reversibility and its higher selectivity for N-type over P/Q type than MVIIA.

Huwentoxin-XVI技術(shù)資料

氨基酸序列:

Cys1-Ile-Gly-Glu-Gly-Val-Pro-Cys8-Asp-Glu-Asn-Asp-Pro-Arg-Cys15-Cys16-Ser-Gly-Leu-Val-Cys21-Leu-Lys-Pro-Thr-Leu-His-Gly-Ile-Trp-Tyr-Lys-Ser-Tyr-Tyr-Cys36-Tyr-Lys-Lys-OH

二硫鍵:Cys1-Cys16, Cys8-Cys21 and Cys15-Cys36

長度 (aa)39

分子式:C196H292N50O56S6

分子量(平均):4437.2 Da

外觀:White lyophilized solid

CAS 號:Not available

來源:Synthetic

純度:> 98%

 

產(chǎn)品信息

貨號

名稱

規(guī)格

N/A

100ug/500ug/1000ug

 

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